oxendolone造句

• Dienogest and oxendolone are unique among the testosterone derivatives in that they are potent antiandrogens.
• The binding affinity of oxendolone for the AR is far lower than that of cyproterone acetate.
• Progestogens that are used as antigonadotropins include chlormadinone acetate, cyproterone acetate, gestonorone caproate, medroxyprogesterone acetate, megestrol acetate, and oxendolone.
• At the AR, oxendolone is not a silent antagonist but is rather predominantly antagonistic with weak agonistic activity; The drug has antigonadotropic properties via its progestogenic actions.
• Although oxendolone is approved for the treatment of BPH in Japan, concerns have been raised about its use for this condition due to poor efficacy seen in clinical trials.